首页> 外国专利> (2S, 3R) - N-(2-((3-piridinil) metr) - 1-azabicyclo 2.2.2 oct-3-il) - 3, 5-difluorohydrazine or an acceptable salt for pharmacodynamics; polymorphism of hydrochloride; pharmacodynamic synthesis; and its use in the treatment of central nervous system diseases such as pain, metabolism, inflammation Alzheimer's disease.

(2S, 3R) - N-(2-((3-piridinil) metr) - 1-azabicyclo 2.2.2 oct-3-il) - 3, 5-difluorohydrazine or an acceptable salt for pharmacodynamics; polymorphism of hydrochloride; pharmacodynamic synthesis; and its use in the treatment of central nervous system diseases such as pain, metabolism, inflammation Alzheimer's disease.

机译:(2S,3R)-N-(2-((3-哌啶子基)metr)-1-氮杂双环[2.2.2] oct-3-il)-3,5-二氟肼或药理学可接受的盐;盐酸盐的多态性药效合成;并用于治疗中枢神经系统疾病,例如疼痛,新陈代谢,炎症,阿尔茨海默氏病。

摘要

Compound (2S, 3R) - N - (2 - (3-pyridinyl) methyl) - 1-azabicyclo [2.2.2] oct - 3 - yl) - 3.5 - diflurobenzamida, polymorphic form of the compoundPharmaceutical Composition and its use for treating or Preventing diseases or Dysfunctions mediated by neuronal nicotinic receptor Alpha 7 such as Pain, metabolic syndrome and inflammationAmong others.
机译:化合物(2S,3R)-N-(2-(3-吡啶基)甲基)-1-氮杂双环[2.2.2]辛基-3-基)-3.5-双氟苯甲酰胺,该化合物的多晶型形式药物组合物及其在治疗中的用途或预防神经元烟碱样受体Alpha 7介导的疾病或功能障碍,例如疼痛,代谢综合征和炎症等。

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