首页> 外国专利> NEW IMIDAZO DERIVATIVES 1,2-a PYRIDINE, METHOD FOR THEIR PRODUCTION, THEIR APPLICATION AS A MEDICINE, PHARMACEUTICAL COMPOSITIONS AND A NEW APPLICATION, PARTICULAR AS INHIBITORS

NEW IMIDAZO DERIVATIVES 1,2-a PYRIDINE, METHOD FOR THEIR PRODUCTION, THEIR APPLICATION AS A MEDICINE, PHARMACEUTICAL COMPOSITIONS AND A NEW APPLICATION, PARTICULAR AS INHIBITORS

机译:新的咪达唑衍生物[1,2-a]吡啶,其制备方法,其在药物中的应用,药物组合物和新的应用,特别是作为抑制剂

摘要

The invention relates to new products of formula (I) in which Ra is H, Hal, aryl or heteroaryl, optionally substituted; Rb is H, Rc, —COORc — CO — Rc or —CO — NRcRd, where Rc is alkyl, cycloalkyl, heterocycloalkyl, aryl and heteroaryl, all optionally substituted; Rd is H, alk or cycloalkyl; moreover, these products are in any isomeric forms and in the form of salts, as medicines, in particular as MET inhibitors.
机译:本发明涉及式(I)的新产物,其中R a是H,Hal,芳基或杂芳基,任选地被取代; Rb为H,Rc,-COORc-CO-Rc或-CO-NRcRd,其中Rc为烷基,环烷基,杂环烷基,芳基和杂芳基,均任选被取代; Rd是H,烷基或环烷基;此外,这些产物呈任何异构形式和盐形式,作为药物,特别是作为MET抑制剂。

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