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New Derivatives of imidazo 1,2-a pyrimidine, its method of preparation, application as Medicines and Pharmaceutical compositions, particularly new use as met inhibitors

机译:咪唑并[1,2-a]嘧啶的新衍生物,其制备方法,在药物和药物组合物中的应用,特别是作为甲胺抑制剂的新用途

摘要

THE INVENTION REFERS TO NEW PRODUCTS OF FORMULA (I): IN WHICH: N = 0.1 OR 2; X REPRESENTS H, HAL, OR ALK; R REPRESENTS H, NH2, NHALK, N (ALK) 2; RA REPRESENTS H; HAL; -O-CYCLLOALKYL; -O-ALKYL, -O-ARYL; -O-HETEROARYL; -NRD (CYCLLOALKYL);-NRD (lessor);-NRD (ARILO)-NRD (heterosexual);1. Aspha cyclopropyl; isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl isopropyl Various forms and salts of these products, mainly as methyl inhibitors
机译:本发明涉及式(I)的新产物:其中:N = 0.1或2; N = 0.1或2。 X代表H,HAL或ALK; R代表H,NH2,NHALK,N(ALK)2; RA代表H; HAL; -O-环烷基; -O-烷基,-O-ARYL; -O-HTEROARYL; -NRD(环烷基);-NRD(出租人);-NRD(ARILO)-NRD(异性恋); 1。沥青;环丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙基异丙醇

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