首页> 外国专利> 1,2,4 - THIADIAZOLE DERIVATIVES, SOME OF WHICH ARE NOVEL AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME FOR TREATING DISORDERS MEDIATED BY MELANOCORTIN RECEPTOR MODULATORS

1,2,4 - THIADIAZOLE DERIVATIVES, SOME OF WHICH ARE NOVEL AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME FOR TREATING DISORDERS MEDIATED BY MELANOCORTIN RECEPTOR MODULATORS

机译:1,2,4-噻二唑衍生物,其中一些是新颖的且包含治疗黑素皮质激素受体调节剂介导的疾病的药物组合物

摘要

The present invention is directed to novel 1,2,4-thiadiazole derivatives of the formula (II) wherein R1, R2 and R4, are ring containing radicals, useful as agonists or antagonists of the melanocortin receptor. More particularly, the compounds of the present invention are useful for the treatment of metabolic, CNS and dermatological disorders.
机译:本发明涉及式(II)的新的1,2,4-噻二唑衍生物,其中R 1,R 2和R 4为含环基团,可用作黑皮质素受体的激动剂或拮抗剂。更特别地,本发明的化合物可用于治疗代谢,CNS和皮肤病学疾病。

著录项

  • 公开/公告号IL161829B

    专利类型

  • 公开/公告日2010-11-30

    原文格式PDF

  • 申请/专利权人 ORTHO-MCNEIL PHARMACEUTICAL INC.;

    申请/专利号IL161829

  • 发明设计人

    申请日2004-05-06

  • 分类号A61K31/429;A61K31/433;A61K31/4439;A61K31/454;A61K31/496;A61K31/541;A61P3/00;A61P3/04;A61P3/10;A61P15/10;A61P17/00;A61P17/10;A61P25/00;A61P27/02;A61P31/10;A61P43/00;C07D285/08;C07D417/02;C07D417/12;

  • 国家 IL

  • 入库时间 2022-08-21 18:06:26

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号