首页> 外国专利> BENZAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, PROCESS FOR THEIR PREPARATION AND USE THEREOF IN THE MANUFACTURE OF MEDICAMENTS AND AS MEDICAMENTS IN THE TREATMENT OF DISEASES ASSOCIATED WITH CANCER

BENZAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, PROCESS FOR THEIR PREPARATION AND USE THEREOF IN THE MANUFACTURE OF MEDICAMENTS AND AS MEDICAMENTS IN THE TREATMENT OF DISEASES ASSOCIATED WITH CANCER

机译:苯甲酰胺衍生物,包含它们的药物组合物,其制备过程及其在药物生产中的用途以及在与癌症有关的疾病治疗中的药物使用

摘要

The invention concerns a compound of the formula (I) wherein Ring A is heterocyclyl; m is 0-4 and each R1 is a group such as hydroxy, halo, trifluoromethyl and cyano; R2 is halo and n is 0-2; and each R4 is a group such as hydroxy, halo, trifluoromethyl and cyano; p is 0-4; and R3 is amino or hydroxy; or pharmaceutically-acceptable salts or in-vivo-hydrolysable ester or amide thereof processes for their preparation, pharmaceutical compositions containing them and their use in the treatment of diseases or medical condions mediated by histone deacetylase.
机译:本发明涉及式(I)的化合物,其中环A是杂环基; m为0〜4,R 1为羟基,卤素,三氟甲基,氰基等基团。 R 2为卤素,n为0-2; R 4为羟基,卤素,三氟甲基,氰基等基团。 p为0-4; R3为氨基或羟基;或它们的药学上可接受的盐或体内可水解的酯或酰胺的制备方法,包含它们的药物组合物及其在治疗由组蛋白脱乙酰基酶介导的疾病或医学病症中的用途。

著录项

  • 公开/公告号IL164373B

    专利类型

  • 公开/公告日2011-02-28

    原文格式PDF

  • 申请/专利号IL164373

  • 申请日2004-10-03

  • 分类号C07D251/14;A61K31/341;A61K31/426;A61K31/427;A61K31/435;A61K31/4365;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/444;A61K31/445;A61K31/4465;A61K31/4525;A61K31/453;A61K31/454;A61K31/47;A61K31/4709;A61K31/4725;A61K31/495;A61K31/4965;A61K31/497;A61K31/505;A61K31/506;A61K31/519;A61K31/53;A61K31/5375;A61K31/5377;A61P7/06;A61P25/14;A61P35/00;A61P43/00;C07D211/34;C07D213/56;C07D213/74;C07D215/12;C07D237/08;C07D239/26;C07D239/42;C07D241/12;C07D241/18;C07D241/20;C07D251/18;C07D277/20;C07D277/24;C07D277/30;C07D295/14;C07D295/155;C07D307/54;C07D401/04;C07D401/06;C07D401/12;C07D403/12;C07D405/06;C07D407/06;C07D409/04;C07D413/04;C07D413/06;C07D417/06;C07D487/04;C07D495/04;

  • 国家 IL

  • 入库时间 2022-08-21 18:06:24

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号