首页> 外国专利> 3 - (2 - {4 - (HEXYLOXYCARBONYLAMINO - IMIINO - METHYL) - PHENYLAMINO - METHYL} - 1 - METHYL - 1H -BENZIMIDAZOL - 5 - CARBONYL) - PYRIDINE - 2 - YL - AMINO - PROPIONIC ACID - ETHYL ESTER METHANE SULPHONATE IN CRYSTAL MODIFICATION I AND II AND ALSO AS A HEMIHYRATE IN ADDITION TO THE USE THEREOF AS A MEDICAMENT.

3 - (2 - {4 - (HEXYLOXYCARBONYLAMINO - IMIINO - METHYL) - PHENYLAMINO - METHYL} - 1 - METHYL - 1H -BENZIMIDAZOL - 5 - CARBONYL) - PYRIDINE - 2 - YL - AMINO - PROPIONIC ACID - ETHYL ESTER METHANE SULPHONATE IN CRYSTAL MODIFICATION I AND II AND ALSO AS A HEMIHYRATE IN ADDITION TO THE USE THEREOF AS A MEDICAMENT.

机译:3-[(2-{[[4-(己基羰基-亚氨基-甲基)-苯胺基]-甲基}-1-甲基-1H-苯并咪唑-5-羰基)-吡啶-2-YL-氨基]-丙酸-乙基结晶形式I和II中的磺酸甲酯磺酸盐,以及除其以外的半水合物,还用作药物。

摘要

The invention relates to the compound 3-[(2-{[4-(hexyloxycarbonylamino-imino-methyl)-phenylamino]-methyl}-1-methyl-1H-benzimidazol-5-carbonyl)-pyridine-2-yl-amino]-propionic acid-ethyl ester methane sulphonate in crystal modifications I and II and also as a hemihyrate in addition to the use thereof as a medicament.
机译:本发明涉及化合物3-[(2-([4-(己氧基氧羰基氨基-亚氨基-甲基)-苯基氨基]-甲基} -1-甲基-1H-苯并咪唑-5-羰基)吡啶-2-基-氨基结晶变体I和II中的]-丙酸-乙酯甲烷磺酸盐,以及除用作药物以外还作为半水合物。

著录项

  • 公开/公告号IL205263A

    专利类型

  • 公开/公告日2011-07-31

    原文格式PDF

  • 申请/专利权人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH;

    申请/专利号IL205263

  • 发明设计人

    申请日2010-04-22

  • 分类号C07D;

  • 国家 IL

  • 入库时间 2022-08-21 18:06:14

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