首页> 外国专利> SUBSTITUTED 4,5,6,7-TETRAHYDROTHIENOPYRIDINES AS KCNQ2/3 MODULATORS FOR TREATING PAIN, EPILEPSY AND URINARY INCONTINENCE.

SUBSTITUTED 4,5,6,7-TETRAHYDROTHIENOPYRIDINES AS KCNQ2/3 MODULATORS FOR TREATING PAIN, EPILEPSY AND URINARY INCONTINENCE.

机译:替代4,5,6,7-四氢噻吩并吡啶类化合物作为KCNQ2 / 3调节剂,用于治疗疼痛,癫痫和尿尿不畅。

摘要

The invention relates to substituted tetrahydrothienopyridines of general formula (1), to a method for the production thereof, to pharmaceutical drugs containing said compounds, and to the use of said compounds for producing pharmaceutical drugs for treating pain, epilepsy, urinary incontinence, anxiety states, addiction, mania, bipolar disorders, migraines, cognitive disorders, dystonia-associated dyskinesias and/or urinary incontinence, where A1 is S, A2 is CRsup14/sup, and A3 is CRsup15/sup; or A1 is CRsup13/sup, A2 is S, and A3 is CRsup15/sup; or A1 is CRsup13/sup, A2 is CRsup14/sup, and A3 is S.
机译:本发明涉及通式(1)的取代的四氢噻吩并吡啶类化合物,其制备方法,含有所述化合物的药物,以及所述化合物在制备用于治疗疼痛,癫痫,尿失禁,焦虑症的药物中的用途。 ,成瘾,躁狂症,躁郁症,偏头痛,认知障碍,肌张力障碍相关的运动障碍和/或尿失禁,其中A1为S,A2为CR 14 ,A3为CR 15 ;或A1为CR 13 ,A2为S,A3为CR 15 ;或A1是CR 13 ,A2是CR 14 和A3是S。

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