首页> 外国专利> THIA-TRIAZA-CYCLOPENTAZULENES AS PI3-KINASES INHIBITORS FOR THE TREATMENT OF CANCER.

THIA-TRIAZA-CYCLOPENTAZULENES AS PI3-KINASES INHIBITORS FOR THE TREATMENT OF CANCER.

机译:噻-三氮杂-环戊二烯酮作为PI3-激酶抑制剂治疗癌症。

摘要

The present invention encompasses compounds of general formula (1) wherein 5 R1 to R3 and X are defined as in claim 1, which are suitable for the treatment of diseases characterised by excessive or abnormal cell proliferation, and the use thereof for preparing a medicament having the above-mentioned properties.
机译:本发明包括通式(1)的化合物,其中5个R 1至R 3和X如权利要求1所定义,其适合于治疗以过度或异常细胞增殖为特征的疾病,及其在制备具有以下特征的药物中的用途:上述特性。

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