首页> 外国专利> N- (2-HYDROXYETHYL) -N-METHYL- 4- (QUINOLIN- 8-YL (1- (THIAZOL-4- YLMETHYL) PIPERIDIN- 4 -YLIDENE) METHYL) BENZAMIDE, THE PROCESS OF MAKING IT AS WELL AS ITS USE FOR THE TREATMENT OF PAIN, ANXIETY AND DEPRESSION

N- (2-HYDROXYETHYL) -N-METHYL- 4- (QUINOLIN- 8-YL (1- (THIAZOL-4- YLMETHYL) PIPERIDIN- 4 -YLIDENE) METHYL) BENZAMIDE, THE PROCESS OF MAKING IT AS WELL AS ITS USE FOR THE TREATMENT OF PAIN, ANXIETY AND DEPRESSION

机译:N-(2-羟基乙基)-N-甲基-4-(喹诺啉-8-基(1-(噻唑-4-基-亚甲基)哌啶-4-亚烷基)甲基)苯甲酰胺的制备方法及其用途用于治疗疼痛,焦虑症和抑郁症

摘要

Disclosed is a N-(2-hydroxyethyl)-N-methyl-4(quinolin-8-yl(1-(thiazole-4-ylmethyl)piperidin-4-ylidene)methyl)benzamide as shown in formula (I) The compound is a delta agonist useful in the treatment of pain, anxiety or depression.
机译:公开了如式(I)所示的N-(2-羟乙基)-N-甲基-4(喹啉-8-基(1-(噻唑-4-基甲基)哌啶-4-亚烷基)甲基)苯甲酰胺。是可用于治疗疼痛,焦虑或抑郁的δ激动剂。

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