首页> 外国专利> PHENYL-{3-(3-(1H-PYRROL-2-YL)-1,2,4OXADIAZOL-5-YLPIPERIDIN-1-YL}-METHANONE DERIVATIVES AND RELATED COMPOUNDS AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS

PHENYL-{3-(3-(1H-PYRROL-2-YL)-1,2,4OXADIAZOL-5-YLPIPERIDIN-1-YL}-METHANONE DERIVATIVES AND RELATED COMPOUNDS AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS

机译:苯甲基-{3-(3-(3-(1H-吡咯-2-基)-[1,2,4]恶二唑-5-基]哌啶-1-基}-甲酮衍生物及相关化合物作为代谢型谷氨酸的正变位调节剂接收器

摘要

The present invention relates to new compounds which are Pyrrole derivatives of formula (I) wherein A, B, P, Q5W, R1 and R2 are defined in the description. Invention compounds are useful in the prevention or treatment of central or peripheral nervous system disorders as well as other disorders modulated by mGluR5 receptors.
机译:本发明涉及新的化合物,它们是式(I)的吡咯衍生物,其中说明书中定义了A,B,P,Q 5 W,R 1和R 2。本发明化合物可用于预防或治疗中枢或周围神经系统疾病以及由mGluR5受体调节的其他疾病。

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