首页> 外国专利> POTENTIATION OF CANCER CHEMOTHERAPY BY 7-(2,5-DIHYDRO-4-IMIDAZO 1,2-APYRINE-3-YL-2,5-DIOXO-IH-PYRROL-3-YL)-9-FLUORO-1,2,3,4 TETRAHYDRO-2-(1-PIPERDINYL-CARBONYL-PYRROLO{3,2,1-JK1,4BENZODIAZEPINE

POTENTIATION OF CANCER CHEMOTHERAPY BY 7-(2,5-DIHYDRO-4-IMIDAZO 1,2-APYRINE-3-YL-2,5-DIOXO-IH-PYRROL-3-YL)-9-FLUORO-1,2,3,4 TETRAHYDRO-2-(1-PIPERDINYL-CARBONYL-PYRROLO{3,2,1-JK1,4BENZODIAZEPINE

机译:7-(2,5-二氢-4-咪唑并[1,2-A]吡咯-3-YL-2,5-二氧羰基-IH-吡咯-3-基)-9-FLUORO-1对癌症的化疗效果,2,3,4四氢-2-(1-哌啶基-羰基-吡咯并{3,2,1-JK] [1,4]苯并二氮杂INE

摘要

A method for treating gastric cancer, ovarian cancer, non-small cell lung cancer, or colorectal cancer in a patient is described, as well as pharmaceutical compositions comprising 7-(2,5-dihydro-4-imidazo[1,2-a]pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4-tetrahydro-2-(1-piperidinyl-carbonyl)-pyrrolo[3,2,1-jk][1,4]benzodiazepine, useful for the method and a process for preparing said compositions.
机译:描述了一种用于治疗患者的胃癌,卵巢癌,非小细胞肺癌或结肠直肠癌的方法,以及包含7-(2,5-二氢-4-咪唑并[1,2-a]的药物组合物。 ]吡啶-3-基-2,5-二氧代-1H-吡咯-3-基)-9-氟-1,2,3,4-四氢-2-(1-哌啶基-羰基)-吡咯[3, 2,1-jk] [1,4]苯并二氮杂,,可用于制备所述组合物的方法和方法。

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