首页> 外国专利> POTENTIATION OF CANCER CHEMOTHERAPY BY 7-(2,5-DIHYDRO-4-IMIDAZO 1,2-APYRINE-3-YL-2,5-DIOXO-IH-PYRROL-3-YL)-9-FLUORO-1,2,3,4 TETRAHYDRO-2-(1-PIPERIDINYL-CARBONYL-PYRROLO3,2,1-JK1,4BENZODIAZEPINE

POTENTIATION OF CANCER CHEMOTHERAPY BY 7-(2,5-DIHYDRO-4-IMIDAZO 1,2-APYRINE-3-YL-2,5-DIOXO-IH-PYRROL-3-YL)-9-FLUORO-1,2,3,4 TETRAHYDRO-2-(1-PIPERIDINYL-CARBONYL-PYRROLO3,2,1-JK1,4BENZODIAZEPINE

机译:7-(2,5-二氢-4-咪唑并[1,2-A]吡啶-3-YL-2,5-二氧-IH-吡咯-3-基)-9-FLUORO-1对癌症的化学治疗作用,2,3,4四氢-2-(1-哌啶基-羰基-吡咯并[3,2,1-JK] [1,4]苯并二氮杂INE

摘要

A method for treating gastric cancer, ovarian cancer, non-small cell lung cancer, or colorectal cancer in a patient is described, as well as pharmaceutical compositions comprising 7-(2,5-dihydro-4-imidazo[ 1, 2-a]pyridine-3-yl-2,5-dioxo-IH-pyrrol-3-yl)-9 tluoro-1,2,3,4 tetrahydro-2- ( l-piperidinyl-carbonyl)-pyrrolo[3,2,1-jk ][I ,4] benzodiazepine, useful for the method and a process for preparing said compositions.
机译:描述了一种用于治疗患者的胃癌,卵巢癌,非小细胞肺癌或结肠直肠癌的方法,以及包含7-(2,5-二氢-4-咪唑并[1、2-a]的药物组合物。 ] pyridine-3-yl-2,5-dioxo-IH-pyrrol-3-yl)-9 tluoro-1,2,3,4 tetrahydro-2-(l-piperidinyl-methoxy)-pyrrolo [3,2, 1-jk] [I,4]苯并二氮杂,可用于制备所述组合物的方法和方法。

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