首页> 外国专利> (E)-N-{3-1-(8-FLUORO-11H-10-OXA-1-AZA-DIBENZO-A,D-CYCLOHEPTEN-5-YLIDENE)-PROPYL-PHENYL }-METHYNSULFON AMIDE AS GLUCOCORTICOID RECEPTOR MODULATOR FOR THE TREATMENT OF RHEUMATOID ARTHRITIS

(E)-N-{3-1-(8-FLUORO-11H-10-OXA-1-AZA-DIBENZO-A,D-CYCLOHEPTEN-5-YLIDENE)-PROPYL-PHENYL }-METHYNSULFON AMIDE AS GLUCOCORTICOID RECEPTOR MODULATOR FOR THE TREATMENT OF RHEUMATOID ARTHRITIS

机译:(E)-N- {3- [1-(8-FLUORO-11H-10-OXA-1-AZA-二苯偶氮-[A,D]-环庚基-5-亚烷基)-丙基]-苯基}-甲基亚磺酰胺作为糖皮质激素受体调节剂,用于治疗类风湿关节炎

摘要

The present invention provides Compound (I) or a pharmaceutically acceptable salt thereof; pharmaceutical compositions comprising Compound (I) in combination with one or more pharmaceutically acceptable carriers, excipients, or diluents; and discloses methods for the treatment of inflammatory and immune disorders comprising administering to a patient in need thereof an effective amount of Compound (I) or a pharmaceutically acceptable salt thereof.
机译:本发明提供了化合物(I)或其药学上可接受的盐;包含化合物(I)与一种或多种药学上可接受的载体,赋形剂或稀释剂组合的药物组合物;公开了治疗炎性和免疫性疾病的方法,包括向有需要的患者施用有效量的化合物(I)或其药学上可接受的盐。

著录项

  • 公开/公告号EP2231676B1

    专利类型

  • 公开/公告日2011-08-31

    原文格式PDF

  • 申请/专利权人 ELI LILLY & COMPANY;

    申请/专利号EP20090701170

  • 申请日2009-01-08

  • 分类号C07D491/04;A61K31/4353;A61P19/02;A61P11/06;

  • 国家 EP

  • 入库时间 2022-08-21 17:56:55

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