首页> 外国专利> USE OF 10-(3R)-1-AZABICYCLO2.2.2OCT-3-YLMETHYL-10H-PHENOTHIAZINE FOR THE PREPARATION OF A DRUG HAVING A SELECTIVE INHIBITION OF MUSCARINIC M1, M2 AND M3 RECEPTORS

USE OF 10-(3R)-1-AZABICYCLO2.2.2OCT-3-YLMETHYL-10H-PHENOTHIAZINE FOR THE PREPARATION OF A DRUG HAVING A SELECTIVE INHIBITION OF MUSCARINIC M1, M2 AND M3 RECEPTORS

机译:使用10-[(3R)-1-氮杂双环[2.2.2] OCT-3-甲基] -10H-苯并噻嗪制备可选择性抑制肌肉M1,M2和M3受体的药物

摘要

Disclosed is a use of 10-[(3R)-1-azabicyclo[2.2.2]oct-3-ylmethyl]-10H-phenothiazine as well as one of its pharmaceutically acceptable salts for the manufacture of a drug to prevent or treat urinary incontinence by selective inhibition of the M1 M2 and M3 muscarinic receptors.
机译:公开了10-[((3R)-1-氮杂双环[2.2.2]辛-3-基甲基] -10H-吩噻嗪及其药学上可接受的盐之一在制备用于预防或治疗尿液的药物中的用途。通过选择性抑制M1 M2和M3毒蕈碱受体实现失禁。

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