首页> 外国专利> LIDOCAINE AS A TRANSFORMER AND PRODUCER OF TRANSFORMED COMPLEXES OF DRUGS DELIVERED IN NANO-DOSAGES USING INJECTION IMPLANTS AS PROLONGED RELEASE DEVICES

LIDOCAINE AS A TRANSFORMER AND PRODUCER OF TRANSFORMED COMPLEXES OF DRUGS DELIVERED IN NANO-DOSAGES USING INJECTION IMPLANTS AS PROLONGED RELEASE DEVICES

机译:利多卡因作为注射剂作为长时间释放装置的纳米剂量药物的转化物和复合物的生产者

摘要

The invention relates to a specific method based on suitable quantities of lidocaine for the transformation of drugs approved by the FDA and COFEPRIS, either in liquid or lyopilised form, producing nano-dosages that do not reduce the effectiveness or the therapeutic effects of the drug, converting same into lidocaine-drug complexes. The transformation method, which results in an end product comprising the fusion of molecules of lidocaine with one or more substances comprising drugs, the prior art and the different methods, techniques and instruments result in the formation of intelligent transformed complexes which can be implanted by means of injection close to the specific receptors, characterised by a release that lasts between 8 and 10 days.
机译:本发明涉及基于适量利多卡因用于转化由FDA和COFEPRIS批准的液体或冻干形式的药物的特定方法,其产生不会降低该药物的有效性或治疗效果的纳米剂量,将其转化为利多卡因-药物复合物。所述转化方法导致最终产物,所述最终产物包括利多卡因分子与一种或多种包含药物的物质融合,现有技术以及不同的方法,技术和仪器导致形成智能转化的复合物,所述复合物可以通过以下方式植入:接近特定受体的注射剂量,其特征在于持续8至10天的释放。

著录项

  • 公开/公告号WO2011145914A1

    专利类型

  • 公开/公告日2011-11-24

    原文格式PDF

  • 申请/专利权人 ZEPEDA FLORES ALEJANDRA;

    申请/专利号WO2011MX00059

  • 发明设计人 ZEPEDA FLORES ALEJANDRA;

    申请日2011-05-16

  • 分类号A61K31/167;

  • 国家 WO

  • 入库时间 2022-08-21 17:18:51

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号