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SULFAMIC ACID ESTER COMPOUNDS USEFUL IN THE INHIBITION OF STEROID SULPHATASE ACTIVITY AND AROMATASE ACTIVITY

机译:用于抑制类固醇硫酸酯酶活性和芳香化酶活性的硫酸酯化合物

摘要

There is provided a compound of Formula (III) or Formula (IV), wherein A is selected from H, OH, halogen and hydrocarbyl D, E and F are each independently of each other an optional linker group; P, Q and R are independently of each other a ring system, wherein R4 and R5 are independently selected from H, alkyl, cycloalkyl, alkenyl, acyl and aryl, or combinations thereof, or together represent alkylene, wherein the or each alkyl or cycloalkyl or alkenyl or optionally contain one or more hetero atoms or groups.
机译:提供了式(III)或式(IV)的化合物,其中A选自H,OH,卤素和烃基D,E和F彼此独立地为任选的连接基团; P,Q和R彼此独立地为环系统,其中R4和R5独立地选自H,烷基,环烷基,烯基,酰基和芳基,或它们的组合,或一起代表亚烷基,其中所述或每个烷基或环烷基或烯基或任选地包含一个或多个杂原子或基团。

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