首页> 外国专利> 1,3-Oxazole-4-carboxamides, 1,3-Thiazole-4-carboxamides, and 1,3-Imidazole-d-carboxamides as Inhibitors of cyclin Dependent kinases

1,3-Oxazole-4-carboxamides, 1,3-Thiazole-4-carboxamides, and 1,3-Imidazole-d-carboxamides as Inhibitors of cyclin Dependent kinases

机译:1,3-恶唑-4-羧酰胺,1,3-噻唑-4-羧酰胺和1,3-咪唑-d-羧酰胺作为细胞周期蛋白依赖性激酶的抑制剂

摘要

Oxazole derivatives are described. The inventive compounds are useful as kinase inhibitors, and may be used in the treatment of cancer, such as prostate cancer, lung cancer, breast cancer, colon cancer, leukemia, CNS cancer, melanoma, ovarian cancer, and renal cancer.
机译:描述了恶唑衍生物。本发明的化合物可用作激酶抑制剂,并且可用于治疗癌症,例如前列腺癌,肺癌,乳腺癌,结肠癌,白血病,CNS癌,黑素瘤,卵巢癌和肾癌。

著录项

  • 公开/公告号US8546400B2

    专利类型

  • 公开/公告日2013-10-01

    原文格式PDF

  • 申请/专利权人 NEOSOME LIFE SCIENCES LLC;

    申请/专利号US201313737328

  • 发明设计人 LAXMAN S. DESAI;SRINIVAS CHITTABOINA;

    申请日2013-01-09

  • 分类号C07D263/48;C07D263/32;C07D417/14;C07D277/593;A61K31/421;A61K31/4178;A61K31/426;A61K31/427;A61P35;A61P1/16;A61P9/10;A61P37/06;

  • 国家 US

  • 入库时间 2022-08-21 16:45:11

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