首页> 外国专利> BIARYL COMPOUNDS AS SERINE PROTEASE INHIBITORS PHARMACEUTICAL COMPOSTIONS, USES, IN VITRO METHODS AND DEVICES COMPRISING SUCH COMPOUNDS

BIARYL COMPOUNDS AS SERINE PROTEASE INHIBITORS PHARMACEUTICAL COMPOSTIONS, USES, IN VITRO METHODS AND DEVICES COMPRISING SUCH COMPOUNDS

机译:含丝氨酸蛋白酶抑制剂的二进制化合物作为制药组合物的用途,体外方法和包含此类化合物的装置

摘要

Compounds of formula (I) are useful as inhibitors of trypsin like serine protease enzymes such as thrombin, factor VIIa, factor Xa, TF/FVIIa, and trypsin. These compounds could be useful to treat and/or prevent clotting disorders, and as anticoagulating agents.
机译:式(I)化合物可用作胰蛋白酶的抑制剂,如丝氨酸蛋白酶,例如凝血酶,VIIa因子,Xa因子,TF / FVIIa和胰蛋白酶。这些化合物可用于治疗和/或预防凝血障碍,并可用作抗凝剂。

著录项

  • 公开/公告号IL222773D0

    专利类型

  • 公开/公告日2012-12-31

    原文格式PDF

  • 申请/专利权人 BIOCRYST PHARMACEUTICALS INC.;

    申请/专利号IL20120222773

  • 发明设计人

    申请日2012-10-30

  • 分类号C07D295/14;A61K31/11;A61K31/192;A61K31/235;A61K31/255;A61K31/27;A61K31/277;A61K31/341;A61K31/352;A61K31/36;A61K31/366;A61K31/381;A61K31/40;A61K31/404;A61K31/416;A61K31/4164;A61K31/4178;A61K31/4184;A61K31/426;A61K31/428;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/453;A61K31/496;A61K31/506;A61K31/535;A61K31/616;A61K31/69;A61K31/695;A61K31/727;A61K38/46;A61K38/48;A61K45;A61P7/02;A61P9/10;A61P29;A61P43;C07C229/38;C07C233/54;C07C233/65;C07C235/84;C07C251/48;C07C255/57;C07C255/58;C07C257/12;C07C257/18;C07C259/18;C07C259/20;C07C271/22;C07C271/64;C07C309/65;C07D207/32;C07D207/337;C07D209/08;C07D213/40;C07D213/55;C07D213/56;C07D213/74;C07D213/75;C07D213/78;C07D213/79;C07D213/80;C07D213/81;C07D213/82;C07D231/56;C07D233/24;C07D233/54;C07D233/61;C07D233/64;C07D235/10;C07D235/14;C07D235/30;C07D235/32;C07D239/14;C07D239/42;C07D239/48;C07D277/20;C07D277/30;C07D277/82;C07D295/16;C07D307/54;C07D311/80;C07D317/46;C07D317/60;C07D317/68;C07D333/24;C07D333/38;C07D405/12;C07D521;

  • 国家 IL

  • 入库时间 2022-08-21 16:41:30

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