首页> 外国专利> USE OF IMIDAZOQUINOLINES FOR THE TREATMENT OF EGFR DEPENDENT DISEASES OR DISEASES THAT HAVE ACQUIRED RESISTANCE TO AGENTS THAT TARGET EGFR FAMILY MEMBERS

USE OF IMIDAZOQUINOLINES FOR THE TREATMENT OF EGFR DEPENDENT DISEASES OR DISEASES THAT HAVE ACQUIRED RESISTANCE TO AGENTS THAT TARGET EGFR FAMILY MEMBERS

机译:使用咪唑并喹啉治疗EGFR依赖性疾病或针对EGFR家族成员的药物已获得耐药性的疾病

摘要

The present invention relates to the use of compounds of formula (I) in the treatment of Epidermal Growth Factor Receptor (EGFR) family members dependent diseases or diseases that have acquired resistance to agents that target EGFR family members, use of said compounds for the manufacture of pharmaceutical compositions for the treatment of said diseases, combinations of said compounds with EGFR modulators for said use, methods of treating said diseases with said compounds and pharmaceutical preparations for the treatment of said diseases comprising said compounds alone or in combination, especially with an EGFR modulator.
机译:本发明涉及式(I)化合物在治疗表皮生长因子受体(EGFR)家族成员依赖性疾病或已获得对靶向EGFR家族成员的药剂的抗性的疾病中的用途,所述化合物在制备中的用途用于治疗所述疾病的药物组合物,用于所述用途的所述化合物与EGFR调节剂的组合,用所述化合物治疗所述疾病的方法以及用于治疗所述疾病的药物制剂,所述药物制剂单独或组合使用所述化合物,尤其是与EGFR调制器。

著录项

  • 公开/公告号EP2182948B1

    专利类型

  • 公开/公告日2013-03-06

    原文格式PDF

  • 申请/专利权人 NOVARTIS AG;

    申请/专利号EP20080786340

  • 申请日2008-07-23

  • 分类号A61K31/444;A61K31/4709;A61K45/06;A61P35;

  • 国家 EP

  • 入库时间 2022-08-21 16:34:16

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