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Composition of solid pharmaceutical preparation containing tacrolimus using self-microemulsifying drug delivery system
Composition of solid pharmaceutical preparation containing tacrolimus using self-microemulsifying drug delivery system
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机译:使用自微乳化药物递送系统的包含他克莫司的固体药物制剂的组合物
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摘要
PURPOSE: A solid formulation composition for oral administration of tacrolimus is provided to improve the bioavailability of tacrolimus without inconvenience. CONSTITUTION: A solid formulation composition for oral administration of tacrolimus contains: a base composition of a self micro-emulsifying drug delivery system containing 30-90 wt% of caproyl caprylic macrogol glyceride as a surfactant, 5-45 wt% of propylene glycol caprylate or triglycerides or a mixture thereof, and 5-60 wt% of diethylene glycol monoethyl ether; 0.1-5.3 weight parts of tacrolimus; and 10-60 parts by weight of dioxy silicone.
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