首页> 外国专利> PROCESS FOR THE ENZYMATIC SYNTHESIS OF (7S) 3,4-DIMETHOXYBICYCLO 4.2.0 OCTA-1,3,5-TRIENE 7-CARBOXYLIC ACID OR ITS ESTERS, AND APPLICATION TO THE SYNTHESIS OF IVABRADIN AND IES SALTS

PROCESS FOR THE ENZYMATIC SYNTHESIS OF (7S) 3,4-DIMETHOXYBICYCLO 4.2.0 OCTA-1,3,5-TRIENE 7-CARBOXYLIC ACID OR ITS ESTERS, AND APPLICATION TO THE SYNTHESIS OF IVABRADIN AND IES SALTS

机译:酶法合成(7S)3,4-二甲氧基双环[4.2.0] OCTA-1,3,5-三烯7-羧酸或其酯的方法及其在合成伊瓦布拉定和IES盐中的应用

摘要

Process for the enzymatic synthesis of the compound of formula (I): in which R represents a hydrogen atom or an alkyl group. Application to the synthesis of ivabradine and its addition salts with a pharmaceutically acceptable acid.
机译:酶促合成式(I)化合物的方法:其中R代表氢原子或烷基。与可药用酸合成伊伐布雷定及其加成盐的应用。

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