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METHOD FOR PRODUCING OPTICALLY ACTIVE BICYCLIC COMPOUND BASED ON ASYMMETRIC CYCLIZATION REACTION
METHOD FOR PRODUCING OPTICALLY ACTIVE BICYCLIC COMPOUND BASED ON ASYMMETRIC CYCLIZATION REACTION
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机译:基于非对称循环反应的光学活性双环化合物的制备方法
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摘要
PROBLEM TO BE SOLVED: To provide a method for optically actively producing bicyclic γ-amino acid derivatives and pharmaceutically acceptable salts thereof, in particular compounds and intermediates thereof having activity as an α2δ ligand.;SOLUTION: Optically active bicyclic compounds are efficiently produced by an asymmetric cyclization reaction.;COPYRIGHT: (C)2014,JPO&INPIT
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