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6,7-dihydro-1,3,4thiadiazolo-3,2-a1,3diazepin derivative and pharmaceutical composition containing the same as neuromuscular blocker or skeletal muscle relaxant, and method for the preparation

机译：6,7-二氢-[1,3,4]噻二唑-[3,2- a ] [1,3]二氮杂pin衍生物和包含与神经肌肉阻滞剂或骨骼肌松弛剂相同的药物组合物，和制备方法

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The present invention relates to a compound of formula 1 and addition salts thereof, a pharmaceutical composition containing the compound, a method for its preparation as well as the use of the compound as neuro-muscular blocker or skeletal muscle relaxant;; wherein each symbol is as defined in the Specification. 展开▼

机译：本发明涉及式1化合物及其加成盐，包含该化合物的药物组合物，其制备方法以及该化合物作为神经肌肉阻滞剂或骨骼肌松弛剂的用途;和其中每个符号如说明书中所定义。展开▼

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公开/公告号US8846665B2

专利类型

公开/公告日2014-09-30

原文格式PDF

申请/专利权人 ADEL S. EL-AZAB;HUSSEIN I. EL-SUBBAGH;KHALID A. AL-RASHOOD;KAMAL E. H. EL-TAHER;MOHAMED A. AL-OMAR;GHADA S. HASSAN;FATMAH A. AL-OMARY;ALAA A. -M. ABDELAZIZ;MOHAMED M. HEFNAWY;
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申请/专利号US201214043401

发明设计人 ADEL S. EL-AZAB;HUSSEIN I. EL-SUBBAGH;KHALID A. AL-RASHOOD;KAMAL E. H. EL-TAHER;MOHAMED A. AL-OMAR;GHADA S. HASSAN;FATMAH A. AL-OMARY;ALAA A. -M. ABDELAZIZ;MOHAMED M. HEFNAWY;
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申请日2012-04-11

分类号A61K31/55;C07D513/04;

国家 US

入库时间 2022-08-21 16:03:19

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