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2-(Substituted-amino)-benzoxazole sulfonamide derivative, its application as medicament, pharmaceutical composition containing thereof and method of in vitro inhibition of retroviral replication

机译:2-(取代的氨基)-苯并恶唑磺酰胺衍生物,其在药物中的应用,包含其的药物组合物以及体外抑制逆转录病毒复制的方法

摘要

The 2-(substituted-amino)-benzoxazole sulfonamide derivative of the general formula (I) and N-oxides, salts, stereoisomeric forms, racemic mixtures or esters thereof. A pharmaceutical application of the derivative, in particular for the inhibition of retrovirus replication. A pharmaceutical composition containing thereof and a method of in vitro inhibition of retroviral replication using the derivative.
机译:通式(I)的2-(取代的氨基)-苯并恶唑磺酰胺衍生物及其N-氧化物,盐,立体异构形式,外消旋混合物或酯。衍生物的药物应用,特别是用于抑制逆转录病毒复制。包含其的药物组合物和使用该衍生物体外抑制逆转录病毒复制的方法。

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