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VITAMIN D DERIVATIVES ACTIVE ON THE VITAMIN D NUCLEAR RECEPTOR, PREPARATION AND USES THEREOF

机译:在维生素D核受体上有活性的维生素D衍生物,制备及其用途

摘要

The invention relates to vitamin D derivatives and their uses, particularly inthepharmaceutical industry. The invention discloses compounds such as of formula(I):(see formula I)having different interesting biological properties, including vitamin Dnuclearreceptor (VDR) agonist activity, as well as therapeutics methods byadministering saidcompounds, in particular for treating cancer, psoriasis, autoimmune diseases,osteodistrophy and osteoporosis. It further relates to pharmaceuticalcompositionscomprising said compounds and methods for preparing the same.
机译:本发明涉及维生素D衍生物及其用途,特别是在的制药业。本发明公开了式的化合物(一世):(参见公式I)具有不同的有趣生物学特性,包括维生素D核受体(VDR)激动剂活性以及治疗方法管理说化合物,特别是用于治疗癌症,牛皮癣,自身免疫性疾病的化合物,骨质疏松症和骨质疏松症。它还涉及药物成分包含所述化合物及其制备方法。

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