首页> 外国专利> 2-3-DIHYDROBENZO 1,4 DIOXIN-2-ILMETIL DERIVATIVES AS ALFA2C ANTAGONISTS FOR USE IN THE TREATMENT OF PERIPHERAL AND CENTRAL NERVOUS SYSTEM DISEASES.

2-3-DIHYDROBENZO 1,4 DIOXIN-2-ILMETIL DERIVATIVES AS ALFA2C ANTAGONISTS FOR USE IN THE TREATMENT OF PERIPHERAL AND CENTRAL NERVOUS SYSTEM DISEASES.

机译:2-3-二氢苯并[1,4]二恶英-2-伊美特尔衍生物作为ALFA2C拮抗剂,用于治疗周围和中枢神经系统疾病。

摘要

Compounds of formula I wherein X, Z, R1-R4, and m are as defined in the claims, exhibit alpha2C antagonistic activity, and are thus useful as alpha2C antagonists. Methods for the treatment of diseases and conditions of the peripheric system and the central nervous system are also disclosed.
机译:其中X,Z,R 1 -R 4和m如权利要求所定义的式I化合物表现出α2 C拮抗活性,因此可用作α2 C拮抗剂。还公开了用于治疗周围系统和中枢神经系统的疾病和状况的方法。

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