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4-imidazolidinones as kv1.5 potassium channel inhibitors

机译:4-咪唑啉酮类化合物作为kv1.5钾通道抑制剂

摘要

The present teachings relate to 4-imidazolidinones of Formula (Ia) or (Ib) which are useful as Kv1.5 potassium channel inhibitors providing atrial-selective antiarrhythmic activity. The present teachings further relate to compositions and methods for treating atrial-selective antiarrhythmia.
机译:本教导涉及式(Ia)或(Ib)的4-咪唑啉酮,其可用作提供心房选择性抗心律不齐活性的Kv1.5钾通道抑制剂。本教导还涉及用于治疗心房选择性抗心律不齐的组合物和方法。

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