PRIORITIES OF PRODUCTION OF THE BUDGET WITH IMPROVED BIOLOGICAL ACTION AND IMPROVED DIALTY, AS CONNECTS FOR PROJECT G (GPCRS) RELATED SUBSTANCES

摘要

The present invention provides prototype_derivatives with improved properties, which can be used as inhibitors of G protein-coupled receptors. Thus, the performance of the treatment under the new compound provides pathological conditions depends on the action of PI alpha theta_beta___953;_uuuuuuuuu The efficiency of G protein coupled receptors.In particular, the compounds of this invention conform to competition and inhibit LHRH receptors. The invention also provides one or more of the original compounds in the medicine as active substances. These agents are particularly suitable for oral use in mammals or humans.