首页> 外国专利> A PROCESS FOR PREPARING FORM A OF (S)-5-METHOXY-2-(4-METHOXY-3,5-DIMETHYL-2- PYRIDINYL)-METHYL SULFINYL1H-BENZIMIDAZOLE MAGNESIUM DIHYDRATE

A PROCESS FOR PREPARING FORM A OF (S)-5-METHOXY-2-(4-METHOXY-3,5-DIMETHYL-2- PYRIDINYL)-METHYL SULFINYL1H-BENZIMIDAZOLE MAGNESIUM DIHYDRATE

机译:(S)-5-甲氧基-2-[[[(4-甲氧基-3,5-二甲基-2-吡啶基)-甲基]亚磺酰基] 1H-苯并咪唑二水合镁的晶型A的制备方法

摘要

A process for preparing Form A of (S) -5-methoxy-2- [ [ (4-methoxy-3, 5-dimethyl-2-pyridinyl) - methyl] sulf inyl] -1 H-benzimidazole magnesium dihydrate, processes for preparing various intermediates useful in the preparation of Form A of (S) -5-methoxy-2- [ [ (4-methoxy-3, 5-dimethyl-2-pyridinyl) -methyl] sulf inyl] -1 H-benzimidazole magnesium dihydrate and a novel polymorphic Form II of 5-methoxy-2- [ [ (4-methoxy-3, 5-dimethyl-2-pyridinyl) -methyl] thio] -1 H-benzimidazole.
机译:(S)-5-甲氧基-2-[[[(4-甲氧基-3,5-二甲基-2-吡啶基)-甲基]硫基] -1 H-苯并咪唑镁二水合物的形式A的制备方法制备可用于制备(S)-5-甲氧基-2-[[[(4-甲氧基-3,5-二甲基-2-吡啶基)-甲基]磺基] -1 H-苯并咪唑镁的形式A的各种中间体二水合物和5-甲氧基-2-[[[(4-甲氧基-3,5-二甲基-2-吡啶基)-甲基]硫代] -1 H-苯并咪唑的新型多晶型物II。

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