首页> 外国专利> AMPHIPHILIC DERIVATIVES OF TRIAZAMACROCYCLE COMPOUNDS, PRODUCTS AND COMPOSITIONS COMPRISING SAME, PROCESSES FOR THEIR SYNTHESIS AND USES THEREOF

AMPHIPHILIC DERIVATIVES OF TRIAZAMACROCYCLE COMPOUNDS, PRODUCTS AND COMPOSITIONS COMPRISING SAME, PROCESSES FOR THEIR SYNTHESIS AND USES THEREOF

机译:三唑类化合物,其产物和组成相同的两亲衍生物,其合成方法及其用途

摘要

The invention relates to amphiphilic derivatives of a triazamacrocyclic compound, as well as to said derivatives as active molecule transporters. The invention also relates to a nanodrug including at least one amphiphilic derivative of a triazamacrocyclic compound and at least one active molecule of a protein such as an antibody, in particular for the treatment of autoimmune diseases or for the treatment of cancer.
机译:本发明涉及三氮杂大环化合物的两亲衍生物,以及涉及作为活性分子转运蛋白的所述衍生物。本发明还涉及一种纳米药物,其包括至少一种三氮杂大环化合物的两亲衍生物和至少一种蛋白质例如抗体的活性分子,特别是用于治疗自身免疫性疾病或用于治疗癌症。

著录项

  • 公开/公告号FR3001217B1

    专利类型

  • 公开/公告日2015-08-14

    原文格式PDF

  • 申请/专利权人 BIOCELLCHALLENGE;

    申请/专利号FR20130000125

  • 申请日2013-01-21

  • 分类号C07D255/02;A61K31/395;A61P35;

  • 国家 FR

  • 入库时间 2022-08-21 14:54:22

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