首页> 外国专利> NOVEL CYCLIC PEPTIDE COMPOUND, PROCESS FOR PRODUCING THE SAME AND INFECTIVE TREATMENT DRUG, ANTIBIOTIC-CONTAINING FRACTS, ANTIBIOTIC AND ANTIBIOTIC MANUFACTURING METHOD, AND ANTIBIOTIC PRODUCING MICROORGANISM

NOVEL CYCLIC PEPTIDE COMPOUND, PROCESS FOR PRODUCING THE SAME AND INFECTIVE TREATMENT DRUG, ANTIBIOTIC-CONTAINING FRACTS, ANTIBIOTIC AND ANTIBIOTIC MANUFACTURING METHOD, AND ANTIBIOTIC PRODUCING MICROORGANISM

机译:新型环肽化合物,生产相同且具有感染力的药物的过程,含抗生素的碎片,抗微生物和抗微生物的制备方法以及产生微生物的微生物

摘要

Provided are: a novel compound having a structure different from that of existing drugs; a novel microorganism capable of producing the novel compound; and further; a novel compound effective to a multiple-drug-resistant bacterium. To provide a novel compound having a high therapeutic effect which can be expected to have a low hurdle for practical realization by selecting an intended compound from many candidate compounds based not only on an antibacterial activity but also on evaluation including a therapeutic effect, a cyclic peptide compound shown by the following formula (1) or a pharmaceutically allowable salt thereof and a microorganism with Accession No. NITE BP-870 or a microorganism mutated naturally or artificially therefrom are provided.
机译:提供:具有不同于现有药物结构的新型化合物;能产生新化合物的新微生物;并进一步;一种对多重耐药细菌有效的新型化合物。通过不仅基于抗菌活性而且还基于包括治疗效果的评价,​​从许多候选化合物中选择所需的化合物,从而提供一种具有高治疗效果的新型化合物,该化合物通过从许多候选化合物中选择所需的化合物,从而可以预期地实现实用化的目标。提供下式(1)所示的化合物或其药学上允许的盐和登录号为NITE BP-870的微生物或从其天然或人工突变的微生物。

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