首页> 外国专利> LONG-CHAIN FATTY ACYL ELONGASE INHIBITOR COMPRISING ARYLSULFONYL DERIVATIVE AS ACTIVE INGREDIENT

LONG-CHAIN FATTY ACYL ELONGASE INHIBITOR COMPRISING ARYLSULFONYL DERIVATIVE AS ACTIVE INGREDIENT

机译:包含芳基磺酰基衍生物作为活性成分的长链脂肪酸酰基转移酶抑制剂

摘要

To provide compounds useful as preventives or remedies for circular systemdisorders, nervous system disorders, metabolic disorders, reproduction systemdisorders,digestive system disorders, neoplasm, infectious diseases, etc., or asherbicides.A long-chain fatty acyl elongase inhibitor comprising, as the activeingredient thereof, a compound or a pharmaceutically-active salt thereof of aformula (I):[Chemical Formula 1](see formula I)[wherein W represents a hydrogen atom, a C1-6 alkyl, etc.; X represents anaryl, a heteroaryl, etc.;n indicates 0 or 1; Z represents a hydrogen atom, a C1-6 alkyl, etc.; A1, A2,A3 and A4 eachindependently represent CH or N].
机译:提供可用作预防或治疗循环系统的化合物疾病,神经系统疾病,代谢疾病,生殖系统疾病,消化系统疾病,肿瘤,传染病等,或除草剂。一种长链脂肪酰基延长酶抑制剂,其包含作为活性成分的其成分,化合物或其药物活性盐公式(I):[化学式1](参见公式I)[其中W表示氢原子,C 1-6烷基等; X代表芳基,杂芳基等;n表示0或1; Z表示氢原子,碳数1〜6的烷基等。 A1,A2,分别为A3和A4独立代表CH或N]。

著录项

  • 公开/公告号CA2722075C

    专利类型

  • 公开/公告日2015-11-24

    原文格式PDF

  • 申请/专利权人 BANYU PHARMACEUTICAL CO. LTD.;

    申请/专利号CA20092722075

  • 申请日2009-04-17

  • 分类号C07D207/48;A61K31/167;A61K31/18;A61K31/197;A61K31/40;A61K31/407;A61K31/4155;A61K31/4184;A61K31/4196;A61K31/437;A61K31/439;A61K31/4439;A61K31/444;A61K31/445;A61K31/454;A61K31/4545;A61K31/4709;A61K31/4965;A61K31/4985;A61K31/4995;A61K31/505;A61K31/506;A61K31/5375;A61K31/5377;A61K31/55;A61P1/16;A61P1/18;A61P3/04;A61P3/06;A61P3/10;A61P3/12;A61P5;A61P9;A61P9/04;A61P9/10;A61P9/12;A61P11;A61P13/12;A61P15/08;A61P17/02;A61P19/02;A61P19/06;A61P27/02;A61P29;A61P31/04;A61P31/10;A61P33;A61P35;A61P43;C07C311/16;C07C317/44;C07D209/52;C07D211/96;C07D213/75;C07D215/38;C07D217/02;C07D231/12;C07D235/14;C07D239/38;C07D241/18;C07D249/12;C07D265/30;C07D295/20;C07D401/04;C07D401/12;C07D401/14;C07D403/12;C07D413/04;C07D413/12;C07D453/06;C07D471/04;C07D487/08;C07D498/04;

  • 国家 CA

  • 入库时间 2022-08-21 14:21:50

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