首页> 外国专利> FOLATE RECEPTOR TARGETED COMPOUND AND PHARMACOLOGICALLY ACCEPTABLE SALTS THEREOF, AND COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT FOR PREVENTION, DIAGNOSIS OR TREATMENT OF CANCER

FOLATE RECEPTOR TARGETED COMPOUND AND PHARMACOLOGICALLY ACCEPTABLE SALTS THEREOF, AND COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT FOR PREVENTION, DIAGNOSIS OR TREATMENT OF CANCER

机译:叶受体靶向的化合物及其药理学可接受的盐,其组成成分与癌症的预防,诊断或治疗相同

摘要

The present invention relates to: a compound for targeting folate receptors, which has a peptide having an amino acid sequence of glycine-glycine-cysteine-glutamate (GGCE) bonded to folic acid, and which can be used for preventing, diagnosing, or treating cancer by specifically bonding to cancer cells having overexpressed folate receptors; or pharmaceutically acceptable salt thereof; and a composition comprising the same as an active component for preventing, diagnosing, or treating cancer.
机译:本发明涉及:一种靶向叶酸受体的化合物,其具有与叶酸结合的具有甘氨酸-甘氨酸-半胱氨酸-谷氨酸(GGCE)的氨基酸序列的肽,并且可用于预防,诊断或治疗。通过与具有过度表达的叶酸受体的癌细胞特异性结合来实现癌症;或其药学上可接受的盐;包含与作为预防,诊断或治疗癌症的活性成分的组合物的组合物。

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