首页> 外国专利> 7-3,5-DIHYDROXY-2-(3-HYDROXY-5-PHENYL-PENT-1-ENYL)-CYCLOPENTYL-N-ETHYL-HEPT-5-ENEAMIDE (BIMATOPROST) IN CRYSTALLINE FORM II, METHODS OF THEREOF OBTAINING AND METHODS FOR APPLICATION THEREOF

7-3,5-DIHYDROXY-2-(3-HYDROXY-5-PHENYL-PENT-1-ENYL)-CYCLOPENTYL-N-ETHYL-HEPT-5-ENEAMIDE (BIMATOPROST) IN CRYSTALLINE FORM II, METHODS OF THEREOF OBTAINING AND METHODS FOR APPLICATION THEREOF

机译：结晶形式II中的7- [3,5-二羟基-2-（3-羟基-5-苯基-戊-1-烯基）-环戊基] -N-乙基-庚-5-乙酰胺（双前体）及其制备方法获得方法及其应用方法

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FIELD: chemistry.;SUBSTANCE: invention relates to novel crystalline form of bimatoprost ((Z)-7-[(1R,2R,3R,5S)-3,5-dihydroxy-2-[(E,3S)-3-hydroxy-5-phenyl-pent-1-enyl]-cyclopentyl]-N-ethyl-hept-5-eneamide), method for thereof obtaining, pharmaceutical composition, containing it, and method for treating ocular hypertension and glaucoma.;EFFECT: novel crystalline form of bimatoprost, possessing higher stability.;8 cl, 7 dwg, 6 tbl

机译：技术领域：本发明涉及比马前列素（（Z）-7-[（1R，2R，3R，5S）-3,5-二羟基-2-[（E，3S）-3-羟基-5-苯基-戊-1-烯基]-环戊基] -N-乙基庚基-5-烯酰胺），其获得方法，包含其的药物组合物以及治疗高眼压和青光眼的方法;效果：比马前列素的新型结晶形式，具有较高的稳定性。; 8 cl，7 dwg，6 tbl

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公开/公告号RU2577546C2

专利类型
公开/公告日2016-03-20

原文格式PDF
申请/专利权人 ALLERGAN INK.;
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申请/专利号RU20120125185
发明设计人 EMBRAS DZHIORDZHI F. (US);KEJRAMI KAJOMARS (US);VU KE (US);
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申请日2010-11-19
分类号C07C405;A61K31/5575;A61P27/06;
国家 RU
入库时间 2022-08-21 14:10:53

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