首页> 外国专利> METHOD FOR SCREENING COMPOUND SPECIFICALLY SUPPRESSING FORMATION OF CAVEOLAE OF CANCER CELLS, SCREENING KIT, VECTOR AND TRANSFORMANT TO BE USED IN KIT, AND METHOD FOR SELECTING PATIENT FOR WHOM MOLECULARLY TARGETED DRUG IS INDICATED

METHOD FOR SCREENING COMPOUND SPECIFICALLY SUPPRESSING FORMATION OF CAVEOLAE OF CANCER CELLS, SCREENING KIT, VECTOR AND TRANSFORMANT TO BE USED IN KIT, AND METHOD FOR SELECTING PATIENT FOR WHOM MOLECULARLY TARGETED DRUG IS INDICATED

机译:指示了用于复合地特别抑制癌细胞的小窝形成的方法,用于该工具中的筛查工具,向量和转化子,以及选择针对谁是分子靶向药物的患者的方法

摘要

Provided is a method for screening a compound that can specifically suppress the formation of caveolae of cancer cells and can inhibit the activity of various RTKs using a single compound all at once. A method for screening a compound specifically suppressing the formation of caveolae of cancer cells wherein the screening method includes a step for bringing a test compound into contact with a system capable of detecting suppression of the binding of Cavin-1 and CAV1 and a step for selecting a compound having activity to suppress the binding of Cavin-1 and CAV1.
机译:本发明提供了一种使用单一化合物一次即可特异性抑制癌细胞小窝形成并抑制各种RTK活性的化合物的筛选方法。筛选特异性抑制癌细胞的小窝形成的化合物的方法,其中筛选方法包括使测试化合物与能够检测Cavin-1和CAV1结合的抑制的系统接触的步骤和选择步骤。具有抑制Cavin-1和CAV1结合的活性的化合物。

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