首页> 外国专利> Crystalline 6-(2-((4-amino-3-(3-hydroxyphenyl)-1H-pyrazolo3,4-Dpyrimidin-1-yl)methyl)-3-(2-chlorobenzyl)-4-0X0-3,4-dihydroquinazolin-5-yl)-N,N-bis(2-methoxyethyl)hex-5-ynamide

Crystalline 6-(2-((4-amino-3-(3-hydroxyphenyl)-1H-pyrazolo3,4-Dpyrimidin-1-yl)methyl)-3-(2-chlorobenzyl)-4-0X0-3,4-dihydroquinazolin-5-yl)-N,N-bis(2-methoxyethyl)hex-5-ynamide

机译:结晶6-(2-(((4-氨基-3-(3-羟基苯基)-1H-吡唑并[3,4-D]嘧啶-1-基)甲基)-3-(2-氯苄基)-4-0X0 -3,4-二氢喹唑啉-5-基)-N,N-双(2-甲氧基乙基)己-5-炔基

摘要

There is provided inter alia 6-(2-((4-amino-3-(3-hydroxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl) methyl)-3-(2-chlorobenzyl)-4-oxo-3,4-dihydroquinazolin-5-yl)-N,N-bis(2-methoxyethyl)hex-5-ynamide in the form of a solid crystalline hydrate and in solid crystalline anhydrous form. There are also provided dry powder pharmaceutical compositions for inhalation containing such solid crystalline forms.
机译:特别提供了6-(2-((4-氨基-3-(3-羟基苯基)-1H-吡唑并[3,4-d]嘧啶-1-基)甲基)-3-(2-氯苄基)固体结晶水合物形式和固体结晶无水形式的-4--4-氧-3,4-二氢喹唑啉-5-基)-N,N-双(2-甲氧基乙基)己-5-炔基。还提供了含有这种固体结晶形式的用于吸入的干粉药物组合物。

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