首页> 外国专利> 1- (5 '- (5- (3,5-dichloro-4-fluorophenyl) -5- (trifluoromethyl) -4,5-dihydroisoxazol-3-yl) -3'h-spiro azetidine crystalline forms -3,1'-isobenzofuran -1-yl) -2- (methylsulfonyl) ethanone

1- (5 '- (5- (3,5-dichloro-4-fluorophenyl) -5- (trifluoromethyl) -4,5-dihydroisoxazol-3-yl) -3'h-spiro azetidine crystalline forms -3,1'-isobenzofuran -1-yl) -2- (methylsulfonyl) ethanone

机译:1-(5'-(5-(3,5-二氯-4-氟苯基)-5-(三氟甲基)-4,5-二氢异恶唑-3-基)-3'h-螺[氮杂环丁烷]晶型-3 ,1'-异苯并呋喃] -1-基)-2-(甲基磺酰基)乙酮

摘要

Patent Summary: "Crystalline forms of 1- (5 '- (5- (3,5-dichloro-4-fluorophenyl) -5- (trifluoromethyl) -4,5-dihydroisoxazol-3-yl) -3 'h-spiro [azetidin-3,1'-isobenzofuran] -1-yl) -2- (methylsulfonyl) ethanone ". The present invention relates to novel crystalline modifications of 1- (5 '- (5- (3,5-dichloro-4-fluorophenyl) -5- (trifluoromethyl) -4,5-dihydroisoxazol-3-yl) -3'h-spiro [azetidin-3,1'-isobenzofuran] -1-yl) -2- (methylsulfonyl) ethanone. The present invention also describes compositions and methods of treating a parasitic infection or infestation in an animal in need thereof. The present invention also relates to processes for producing crystalline forms.
机译:专利摘要:“ 1-(5'-(5-(3,5-二氯-4-氟苯基)-5-(三氟甲基)-4,5-二氢异恶唑-3-基)-3'h-螺环的结晶形式[氮杂环丁烷-3,1'-异苯并呋喃] -1-基)-2-(甲基磺酰基)乙酮。本发明涉及1-(5'-(5-(3,5-二氯-4-氟苯基)-5-(三氟甲基)-4,5-二氢异恶唑-3-基)-3'h的新型晶体修饰-螺环[氮杂环丁烷-3,1'-异苯并呋喃] -1-基)-2-(甲基磺酰基)乙酮。本发明还描述了在需要其的动物中治疗寄生虫感染或侵扰的组合物和方法。本发明还涉及生产结晶形式的方法。

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