首页> 外国专利> PRODUCTS OF 7-(PETROYL-AMINO)-6,7,8,9-THIRD BUDGET1,2-aOXIC INDOLD AND THEIR USE AS CHARACTERISTICS OF THE SUBSTANCE OF PROGRAMME D2

PRODUCTS OF 7-(PETROYL-AMINO)-6,7,8,9-THIRD BUDGET1,2-aOXIC INDOLD AND THEIR USE AS CHARACTERISTICS OF THE SUBSTANCE OF PROGRAMME D2

机译:7-(邻苯二甲酰氨基)-6,7,8,9-第三预算[1,2-a]氧的产物及其作为程序D2物质特征的用途

摘要

The present invention relates to the formula (I) of a derivative (e__alpha p_lambda-7-6, 7, 8, 9-amino) - _____delta_ [1, 2-a] _delta lambda_acetic acid, in which R1, R2, R3 and R4 PI P p__ In describing and using them as prostaglandin leukotriene receptors, especially leukotriene prostaglandin D2 receptors;A prostaglandin-mediated, containing uniformity in the eyes of pharmaceutical compositions for the treatment of various diseases and disorders. In this way, its preparation method.
机译:本发明涉及衍生物(e_αp_lambda-7-6、7、8、9-氨基)-____ delta_ [1、2-a]_deltaλ_乙酸的式(I),其中R1,R2,R3和R4 PI P p__在描述和用作前列腺素白三烯受体,特别是白三烯前列腺素D2受体时;由前列腺素介导,在药物组合物中具有均匀性,可用于治疗各种疾病和病症。这样,就是其制备方法。

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