首页> 外国专利> MEGLUMINE SALT OF 2-((1R,4R)-4-(4-(5-(BENZOXAZOL-2-YLAMINO)PYRIDIN-2-YL)PHENYL)CYCLOHEXYL)ACETIC ACID AND A CRYSTALLINE FORM THEREOF AND THEIR USE AS DGAT1 INHIBITORS

MEGLUMINE SALT OF 2-((1R,4R)-4-(4-(5-(BENZOXAZOL-2-YLAMINO)PYRIDIN-2-YL)PHENYL)CYCLOHEXYL)ACETIC ACID AND A CRYSTALLINE FORM THEREOF AND THEIR USE AS DGAT1 INHIBITORS

机译:2-((1R,4R)-4-(4-(5-(BENZOXAZOL-2-YLAMINO)PYRIDIN-2-YL)Phenylhecyheylyl)acetic acid和结晶形式的葡甲胺盐及其作为DGAT1抑制剂的用途

摘要

The present invention relates to a meglumine salt of 2-((1R,4R)-4-(4-(5-(benzo[d]oxazol-2-ylamino)pyridin-2-yl)phenyl)cyclohexyl)acetic acid of Formula (I) and a crystalline form thereof and their use in the treatment or prevention of a condition or a disorder associated with DGAT1 activity in animals, particularly humans.
机译:本发明涉及2-((1R,4R)-4-(4-(5-(苯并[d]恶唑-2-基氨基)吡啶-2-基)苯基)环己基)乙酸的葡甲胺盐。式(I)及其结晶形式及其在治疗或预防动物,特别是人中与DGAT1活性有关的病症或病症中的用途。

著录项

  • 公开/公告号EA027688B1

    专利类型

  • 公开/公告日2017-08-31

    原文格式PDF

  • 申请/专利权人 NOVARTIS AG;

    申请/专利号EA20150091300

  • 申请日2014-01-10

  • 分类号C07D413/12;A61K31/4439;A61P3/04;A61P3/10;

  • 国家 EA

  • 入库时间 2022-08-21 13:39:12

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