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1,3-OXAZOLIDINE OR 1,3-OXAZINANE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS

机译:1,3-恶唑烷或1,3-恶嗪烷类化合物作为食欲素受体拮抗剂

摘要

A heteroaromatic methyl cyclic amine derivative represented by formula (IA) or a pharmaceutically acceptable salt thereof is useful for treatment or prophylaxis of diseases such as sleep disorder, depression, anxiety disorder, panic disorder, schizophrenia, drug dependence, Alzheimer's disease, Parkinson's disease, Huntington's disease, eating disorder, cephalalgia, hemicrania, pain, digestive diseases, epilepsy, inflammation, immune-related diseases, endocrine-related diseases and hypertension, on the basis of an orexin (OX) receptor antagonist activity.
机译:由式(IA)表示的杂芳族甲基环胺衍生物或其药学上可接受的盐可用于治疗或预防疾病,例如睡眠障碍,抑郁症,焦虑症,恐慌症,精神分裂症,药物依赖性,阿尔茨海默氏病,帕金森氏病,亨廷顿舞蹈症,进食障碍,头痛,半脑膜炎,疼痛,消化系统疾病,癫痫病,炎症,免疫相关疾病,内分泌相关疾病和高血压,取决于食欲素(OX)受体拮抗剂的活性。

著录项

  • 公开/公告号HRP20161797T1

    专利类型

  • 公开/公告日2017-02-24

    原文格式PDF

  • 申请/专利权人 TAISHO PHARMACEUTICAL CO. LTD;

    申请/专利号HR2016P001797T

  • 申请日2016-12-27

  • 分类号C07D413/14;A61K31/4439;A61K31/5355;A61P1/04;A61P1/14;A61P3;A61P9/12;A61P25/06;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/36;A61P29;A61P37/02;

  • 国家 HR

  • 入库时间 2022-08-21 13:39:07

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