首页> 外国专利> (4-((3R,4R)-3-METHOXYTETRAHYDRO-PYRAN-4-YLAMINO)PIPERIDIN-1-YL)(5-METHYL-6-(((2R,6S)-6-(P-TOLYL)TETRAHYDRO-2H-PYRAN-2-YL)METHYLAMINO)PYRIMIDIN-4YL)METHANONE CITRATE

(4-((3R,4R)-3-METHOXYTETRAHYDRO-PYRAN-4-YLAMINO)PIPERIDIN-1-YL)(5-METHYL-6-(((2R,6S)-6-(P-TOLYL)TETRAHYDRO-2H-PYRAN-2-YL)METHYLAMINO)PYRIMIDIN-4YL)METHANONE CITRATE

机译:(4-(((3 R ,4 R ))-3-甲氧基四氢吡喃-吡喃-4-基氨基)哌啶-1-基)(5-甲基-6-( ((2 R ,6S)-6-(对-甲苯基)四氢-2H-吡喃-2-基)甲氨基)嘧啶-4YL)柠檬酸甲酮酯

摘要

The invention provides a salt of a tetrahydropyranylmethylaminopyrimidine amide, such as the citrate salt of (4-((3R,4R)-3-methoxytetrahydropyran-4-ylamino)piperidin-l-yl)(5-methyl-6-(((2R,6S)-6-(p-tolyl)tetrahydro-2H-pyran-2-yl)methylamino)pyrimidin-4-yl)methanone, pharmaceutical compositions containing the same, processes for preparing the same, and methods of medical treatment using the same.
机译:本发明提供了四氢吡喃基甲基氨基嘧啶酰胺的盐,例如(4-((3R),4R)-3-甲氧基四氢吡喃-4-基氨基)的柠檬酸盐。哌啶-1-基)(5-甲基-6-((((2 R ,6 S) -6-(对甲苯基)四氢-2H-吡喃- 2-基)甲基氨基)嘧啶-4-基)甲酮,含有该基团的药物组合物,其制备方法以及使用其的药物治疗方法。

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