首页> 外国专利> ADDITION SALTS OF N-4-(4-{(1S)-1-(5-METHYL-4-OXO-3-PHENYL-3,4-DIHYDROPYRROLO2,1-F1,2,4TRIAZIN-2-YL)ETHYLAMINO}-7H-PYRROLO2,3-DPYRIMIDIN-5-YL)-1H-INDOL-6-YLSULFAMIDE

ADDITION SALTS OF N-4-(4-{(1S)-1-(5-METHYL-4-OXO-3-PHENYL-3,4-DIHYDROPYRROLO2,1-F1,2,4TRIAZIN-2-YL)ETHYLAMINO}-7H-PYRROLO2,3-DPYRIMIDIN-5-YL)-1H-INDOL-6-YLSULFAMIDE

机译:N- [4-(4-{[(1S)-1-(5-Methylyl-4-OXO-3-Phenyl-3,4-DIHYDROPYYROROROLO [2,1-F] [1,2,4]的附加盐]三嗪-2-基)乙基]酰胺} -7H-吡咯并[2,3-D]嘧啶基-5-基)-1H-吲哚6-基]硫

摘要

The present invention is directed to crystalline addition salts of (I) N-[4-(4-{[(1S)-1-(5-methyl-4-oxo-3-phenyl-3,4-dihydropyrrolo[2,1- f][1,2,4]triazin-2-yl)ethyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-5-yl) -1 H-indol-6-yl]sulfamide with sulfonic acid derivatives, chosen from methanesulfonic acid, ethanesulfonic acid and benzenesulfonic acid, or pharmaceutically acceptable solvates thereof.
机译:本发明涉及(I)N- [4-(4-{[((1S)-1-(5-甲基-4-氧代-3-苯基-3,4-二氢吡咯并[2, 1-f] [1,2,4]三嗪-2-基)乙基]氨基} -7H-吡咯并[2,3-d]嘧啶-5-基)-1 H-吲哚-6-基]磺酰胺与选自甲磺酸,乙磺酸和苯磺酸的磺酸衍生物,或其药学上可接受的溶剂化物。

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