首页> 外国专利> 1-5'-5-35--4--5--45--3--3'H--31'--1--2- CRYSTALLINE FORMS OF 1-5'-5-35-DICHLORO-4-FLUOROPHENYL-5-TRIFLUOROMETHYL-45-DIHYDROISOXAZOL-3-YL-3'H-SPIROAZETIDINE-31'-ISOBENZOFURAN-1-YL-2-METHYLSULFONYLETHANONE

1-5'-5-35--4--5--45--3--3'H--31'--1--2- CRYSTALLINE FORMS OF 1-5'-5-35-DICHLORO-4-FLUOROPHENYL-5-TRIFLUOROMETHYL-45-DIHYDROISOXAZOL-3-YL-3'H-SPIROAZETIDINE-31'-ISOBENZOFURAN-1-YL-2-METHYLSULFONYLETHANONE

机译:1-5'-5-35- 1-5'-5-35--4--5--45--3--3'H-[-31'-]-1--2-晶体形式二氯4-氟代苯基-5-三氟甲基-45-二氢异恶唑-3-基-3'H-螺[氮杂环丁烷-31'-异苯并呋喃] -1-基-2-甲基丁二酮

摘要

The present invention relates to a process for the preparation of 1- (5 ''- (5- (3,5-dichloro-4-fluorophenyl) -5- (trifluoromethyl) -4,5-dihydroisooxazole- -3''H-spiro [azetidine-3,1''-isobenzofuran] -l-yl) -2- (methylsulfonyl) ethanone. The present invention also describes compositions and methods for treating parasitic infections or intravital infections in an animal in need of such treatment. The present invention also relates to a method of producing a crystalline form.
机译:本发明涉及制备1-(5′′-(5-(3,5-二氯-4-氟苯基)-5-(三氟甲基)-4,5-二氢异恶唑--3″ H的方法-螺环[氮杂环丁烷-3,1”-异苯并呋喃] -1-基)-2-(甲磺酰基)乙酮本发明还描述了用于治疗需要这种治疗的动物中的寄生虫感染或玻璃体内感染的组合物和方法。本发明还涉及生产结晶形式的方法。

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