首页> 外国专利> (2S, 5R) -7-oxo-6-sulfooxy-2-((3R) -piperidine-3-carbonyl) -hydrazinocarbonyl -1,6-diaza-bicyclo 3.2.1 octane Process for preparation

(2S, 5R) -7-oxo-6-sulfooxy-2-((3R) -piperidine-3-carbonyl) -hydrazinocarbonyl -1,6-diaza-bicyclo 3.2.1 octane Process for preparation

机译:(2S,5R)-7-氧代-6-磺氧基-2-[(((3R)-哌啶-3-羰基)-肼基羰基] -1,6-二氮杂双环[3.2.1]辛烷的制备方法

摘要

A process for preparation of (2S,5R)-7-oxo-6-sulphooxy-2-[((3R)-piperidine-3-carbonyl)-hydrazino carbonyl]-1,6-diaza-bicyclo[3.2.1]octane of Formula (I) is disclosed which is comprising reacting a compound of Formula (II) with a compound of Formula (III) to obtain a compound of Formula (IV). Crystalline compounds of Formula (I) are claimed.
机译:(2S,5R)-7-氧代-6-磺氧基-2-[(((3R)-哌啶-3-羰基)-肼基羰基] -1,6-二氮杂双环[3.2.1]的制备方法公开了式(I)的辛烷,其包括使式(II)的化合物与式(III)的化合物反应以获得式(IV)的化合物。要求保护式(I)的结晶化合物。

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