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CRYSTAL FORM OF BROMODOMAIN PROTEIN INHIBITOR DRUG, PREPARATION METHOD AND USE THEREOF

机译:溴蛋白抑制剂的结晶形式,制备方法及其用途

摘要

The present disclosure relates to novel crystalline forms of a bromodomain protein inhibitor 2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxyquinazolin-4(3H)-one and processes for preparation and use thereof, relating to pharmaceutical industry. Form CS2, Form CS8, Form CS13, Form CS20, Form CS1, Form CS7, Form CS9, Form CS11 and Form CS4 of the present disclosure can be used for preparing drugs treating cardiovascular, cholesterol or lipid-related disorders.
机译:本公开涉及溴结构域蛋白抑制剂2- [4-(2-羟基乙氧基)-3,5-二甲基苯基] -5,7-二甲氧基喹唑啉-4(3H)-的新型晶型及其制备和用途。 ,与制药业有关。本公开的形式CS2,形式CS8,形式CS13,形式CS20,形式CS1,形式CS7,形式CS9,形式CS11和形式CS4可用于制备治疗心血管,胆固醇或脂质相关疾病的药物。 <图像文件=“ IMGA0001.GIF” he =“ 59” imgContent =“ chem” imgFormat =“ GIF” wi =“ 93” />

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