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PRODUCTION METHOD FOR NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND INTERMEDIATE OF SAID NITROGEN-CONTAINING HETEROCYCLIC COMPOUND

机译:含氮杂环化合物的生产方法以及所述的含氮杂环化合物的中间体

摘要

An object of the present invention is to provide a method for industrially manufacturing a nitrogen-containing heterocyclic compound which shows excellent FLT3 inhibitory activity and is useful as a pharmaceutical active ingredient of pharmaceutical products. The present invention provides a manufacturing method of a compound represented by General Formula [14] or a salt thereof (in the formula, R 1 represents a C 1-6 alkyl group which may be substituted; and R 8 represents a leaving group or the like).
机译:本发明的目的是提供一种工业生产含氮杂环化合物的方法,该化合物显示出优异的FLT3抑制活性,并可用作药物的药物活性成分。本发明提供了由通式[14]表示的化合物或其盐(式中,R 1表示可被取代的C 1-6烷基; R 8表示离去基或喜欢)。

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