首页> 外国专利> COMPOUND HAVING TYROSINE PROTEIN KINASE JAK1- OR JAK2-INHIBITTION AND DEGRADATION ACTIVITY

COMPOUND HAVING TYROSINE PROTEIN KINASE JAK1- OR JAK2-INHIBITTION AND DEGRADATION ACTIVITY

机译:具有酪氨酸蛋白激酶JAK1或JAK2抑制和降解活性的化合物

摘要

The present invention provides a compound having tyrosine protein kinase JAK1- or JAK2-inhibittion and degradation activity. Specifically, the present invention provides a compound as represented by the following formula I, wherein the definition of each group is as stated in the description. The compound provided by the present invention has excellent JAK1- or JAK2-inhibittion and degradation activity, and can be used for preparing drugs for treatment of JAK1- or JAK2-related diseases.
机译:本发明提供了具有酪氨酸蛋白激酶JAK1或JAK2抑制和降解活性的化合物。具体地,本发明提供由下式I表示的化合物,其中每个基团的定义如说明书中所述。本发明提供的化合物具有优异的JAK1或JAK2抑制和降解活性,可用于制备治疗JAK1或JAK2相关疾病的药物。

著录项

  • 公开/公告号WO2019042442A1

    专利类型

  • 公开/公告日2019-03-07

    原文格式PDF

  • 申请/专利权人 SHANGHAI MEIZER PHARMACEUTICALS CO. LTD.;

    申请/专利号WO2018CN103707

  • 发明设计人 SHU YONGZHI;

    申请日2018-09-02

  • 分类号C07D487/04;A61K31/519;A61P35;A61P37/06;A61P19/02;A61P17/06;A61P17;A61P11/06;A61P3/10;A61P1/04;A61P1;A61P25/28;

  • 国家 WO

  • 入库时间 2022-08-21 11:56:20

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