, ;which is the thrombin direct inhibitor, as well as to its production and application method.;EFFECT: ensuring the biologically active substance, the thrombin inhibitor, oral administration possibility, and at that preserving its specific pharmacological activity as the anticoagulant.;4 cl, 1 dwg, 5 tbl"/> 4-AMINO-1-{2-3-METHYL-5-(BENZENESULFONYLOXYPHENOXYETHYL}-PYRIDIUM CHLORIDE SUBSTANCE, HAVING THE BIOLOGICALLY ACTIVE AGENT PROPERTIES, INFLUENCING THE MAMMALS BLOOD COAGULABILITY NATURALLY RUNNING PROCESSES, ANTICOAGULANT ON ITS BASIS AND ITS OBTAINING METHOD BY CHEMICAL SYNTHESIS
首页> 外国专利> 4-AMINO-1-{2-3-METHYL-5-(BENZENESULFONYLOXYPHENOXYETHYL}-PYRIDIUM CHLORIDE SUBSTANCE, HAVING THE BIOLOGICALLY ACTIVE AGENT PROPERTIES, INFLUENCING THE MAMMALS BLOOD COAGULABILITY NATURALLY RUNNING PROCESSES, ANTICOAGULANT ON ITS BASIS AND ITS OBTAINING METHOD BY CHEMICAL SYNTHESIS

4-AMINO-1-{2-3-METHYL-5-(BENZENESULFONYLOXYPHENOXYETHYL}-PYRIDIUM CHLORIDE SUBSTANCE, HAVING THE BIOLOGICALLY ACTIVE AGENT PROPERTIES, INFLUENCING THE MAMMALS BLOOD COAGULABILITY NATURALLY RUNNING PROCESSES, ANTICOAGULANT ON ITS BASIS AND ITS OBTAINING METHOD BY CHEMICAL SYNTHESIS

机译:4-氨基1- {2- [3- [3-甲基-5-(苯并磺酰氧基)苯氧基]乙基]-吡啶鎓氯化物,具有生物活性剂特性,影响哺乳动物血液的自然运行过程的可凝结性,抗氧化剂及其基础。化学合成方法

摘要

FIELD: chemistry.;SUBSTANCE: group of inventions relates to the 4-amino-1-{2-[3-methyl-5-(benzenesulfonyloxy]phenoxy]ethyl}-pyridium chloride, having the structural formula ; , ;which is the thrombin direct inhibitor, as well as to its production and application method.;EFFECT: ensuring the biologically active substance, the thrombin inhibitor, oral administration possibility, and at that preserving its specific pharmacological activity as the anticoagulant.;4 cl, 1 dwg, 5 tbl
机译:发明领域本发明涉及具有结构式的4-氨基-1- {2- [3-甲基-5-(苯磺酰氧基]苯氧基]乙基}-吡啶鎓氯化物。 ,这是凝血酶直接抑制剂,及其生产和使用方法。 ;效果:确保具有生物活性物质,凝血酶抑制剂,口服给药的可能性,并保持其特定的药理活性作为抗凝剂。; 4 cl,1 dwg,5 tbl

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