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NOVEL PROCESS FOR THE PREPARATION OF DIPEPTIDYL PEPTIDASE-4 (DPP-4) ENZYME INHIBITOR

机译:二肽基肽酶-4(DPP-4)酶抑制剂的制备新工艺

摘要

The present invention relates to a novel and improved process for the preparation of Sitagliptin of Formula (I) and its pharmaceutically acceptable salts. The present invention also relates to novel intermediates and process for the preparation of intermediates used in the preparation of Sitagliptin.
机译:本发明涉及制备式(I)西格列汀及其药学上可接受的盐的新颖且改进的方法。本发明还涉及新颖的中间体和用于制备西他列汀的中间体的制备方法。

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