首页> 外国专利> COMPOSITION COMPRISING ETHYL VANILLIN AS EFFECTIVE INGREDIENT FOR EXHIBITING EFFECT OF MUSCLE STRENGTHENING, MUSCLE ENHANCEMENT, MUSCLE DIFFERENTIATION, MUSCLE REGENERATION, OR SARCOPENIA SUPPRESSION

COMPOSITION COMPRISING ETHYL VANILLIN AS EFFECTIVE INGREDIENT FOR EXHIBITING EFFECT OF MUSCLE STRENGTHENING, MUSCLE ENHANCEMENT, MUSCLE DIFFERENTIATION, MUSCLE REGENERATION, OR SARCOPENIA SUPPRESSION

机译:包含乙基香兰素作为有效成分的组合物,可显示增强肌肉,增强肌肉,分化肌肉,再生肌肉或抑制肌肉发达的功效

摘要

The present invention relates to a composition comprising ethyl vanillin or a pharmaceutically acceptable salt thereof as an effective ingredient for preventing or treating muscle disease or for improving a muscle function. Having the capability of upregulating the expression of a protein associated with muscle protein synthesis and muscle mass increase in myocytes and downregulating at an mRNA level the expression of an enzyme involved in muscle protein degradation, ethyl vanillin can exhibit effects of muscle differentiation, muscle regeneration, and muscle strengthening through an increase in muscle mass against muscle diseases attributed to muscle function decrease, muscle consumption, or muscle degradation and can suppress sarcopenia. Thus, ethyl vanillin can be used for preventing or treating muscle diseases or for promoting muscle differentiation, muscle regeneration and muscle strengthening, muscle mass increase, or muscle generation or for improving muscle function.
机译:本发明涉及一种包含乙基香兰素或其药学上可接受的盐作为预防或治疗肌肉疾病或改善肌肉功能的有效成分的组合物。乙基香兰素具有上调与肌肉蛋白质合成和肌细胞中肌肉质量增加相关的蛋白质表达的能力,并在mRNA水平上下调参与肌肉蛋白质降解的酶的表达的能力,因此可以发挥肌肉分化,肌肉再生,通过增加肌肉质量来抵抗因肌肉功能下降,肌肉消耗或肌肉退化引起的肌肉疾病,从而抑制肌肉减少症。因此,乙基香兰素可用于预防或治疗肌肉疾病或用于促进肌肉分化,肌肉再生和肌肉增强,肌肉质量增加或肌肉生成或用于改善肌肉功能。

著录项

  • 公开/公告号US2020170964A1

    专利类型

  • 公开/公告日2020-06-04

    原文格式PDF

  • 申请/专利号US201816631761

  • 发明设计人 TAE SUN PARK;

    申请日2018-07-17

  • 分类号A61K31/11;A23L33/10;A23K20/111;A61P21/04;A61P21/06;

  • 国家 US

  • 入库时间 2022-08-21 11:20:41

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